Drug Metabolism And Pharmacokinetics Drug metabolism and pharmacokinetics (DMPK) is a core discipline in drug development that considers the biotransformation of a drug compound and other pharmacokinetic properties to assess drug safety. DMPK, or commonly referred to as DMPK, is a scientific discipline within drug discovery, dealing with safety and efficacy evaluation of drug candidates before entering clinical trials. https://www.nebiolab.com/drug-metabolism-and-pharmacokinetics-dmpk/